3-氨基香豆素及其衍生物代表了有机合成中一类重要的多任务和多功能支架。因此，3-氨基香豆素的合成及其合成应用在有机化学和药物化学领域具有巨大的影响，因为这类化合物表现出的各种生物活性以及它们的天然存在。由于所述支架中存在氨基和烯胺碳，3-氨基香豆素的化学反应性更为深刻。本综述的目的是关注不同的合成方法，用于合成 3-氨基香豆素衍生物及其生物学评价和荧光研究。

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3-Aminocoumarins and their derivatives represent an important class of a multi-tasking and multi-functional scaffold in organic synthesis. So, the synthesis of 3-aminocoumarins and their synthetic applicability have an immense impact in the field of organic and pharmaceutical chemistry due to various biological activities displayed by such class of compounds as well as due to their natural occurrences. The chemical reactivity of 3-aminocoumarins is more profound due to the presence of an amino group as well as enamine carbon in the described scaffold. The objective of this present review was to focus on different synthetic methodologies, for the synthesis of 3-aminocoumarin derivatives and their biological evaluation and fluorescence study.